噻氯匹定抑制劑CYC116 is a potent inhibitor of Aurora A/B with Ki of 8.0 nM/9.2 nM, is less potent to VEGFR2 (Ki of 44 nM), with 50-fold greater potency than CDKs, not active against PKA, Akt/PKB, PKC, no effect on GSK-3α/β, CK2, Plk1 and SAPK2A. Phase 1.
| 產(chǎn)品名稱： | 噻氯匹定 | ||
| 英文名： | CYC116 | ||
| CAS NO.： | 693228-63-6 | ||
| 分子式： | C18H20N6Os | ||
| 分子量： | 368.456001281738 | ||
| 產(chǎn)品品牌： | targetmol | ||
| 產(chǎn)品規(guī)格： | 2mg | ||
