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GSK J1
貨號(hào):T6847
產(chǎn)品名稱: GSK J1
英文名: GSK J1
CAS NO.: 1373422-53-7
分子式: C22H23N5O2
分子量: 389.450324296951
產(chǎn)品品牌: targetmol
產(chǎn)品規(guī)格: 5mg
GSK J1
GSK J1抑制劑GSK-J1 is a highly potent H3K27 histone demethylase inhibitor with IC50 of 28 nM and 53 nM in cell-free assays for JMJD3 (KDM6B) and UTX (KDM6A), respectively, >10-fold selectivity over other tested demethylases.